Pechmann reaction promoted by boron trifluoride dihydrate.

نویسندگان

  • Edmont V Stoyanov
  • Jochen Mezger
چکیده

The Pechmann reaction of substituted phenols 1a-e with methyl acetoacetate (2) can be activated by boron trifluoride dihydrate (3) to give the corresponding 4-methyl- coumarin derivatives 4a-e in excellent yield (98-99 %).

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عنوان ژورنال:
  • Molecules

دوره 10 7  شماره 

صفحات  -

تاریخ انتشار 2005